

HY-168641 · 5 mg
MedChemExpress · Cat: HY-168641
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medchemexpress.com/protac-hif-1%CE%B1-degrader-1.htmlDescription
PROTAC HIF-1? degrader-1 compound V2 is a potent hypoxia-inducible factor-1? HIF-1? PROTAC degrader with an IC50 value of 7.54 AAasAasAAmuM. PROTAC HIF-1? degrader-1 shows anti-proliferative activity. PROTAC HIF-1? degrader-1 decreases the HIF-1? protein expression. PROTAC HIF-1? degrader-1 induces apoptosis. Pink: ligand for target protein HY-111387 ; black: linker HY-W013731 ; Blue: E3 ligase ligand HY-112078 .







