

HY-157805 · 50 mg
MedChemExpress · Cat: HY-157805
Reach 3+ verified distributors
Manufacturer product page
medchemexpress.com/protac-sars-cov-2-mpro-degrader-2.htmlDescription
PROTAC SARS-CoV-2 Mpro degrader-2 Compound 6 is a potent PROTAC degrader of SARS-CoV-2 Mpro. PROTAC SARS-CoV-2 Mpro degrader-2 has broad-spectrum antiviral activity against CoVs, including SARS-CoV-2 EC50 = 10.8 ?M , HCoV-OC43 EC50 = 1.6 ?M and HCoV-229E EC50 = 6.5 ?M . PROTAC SARS-CoV-2 Mpro degrader-2 exhibits potent activity against SARS-CoV-2 in Calu-3 cells, with an EC50 of 0.89 ?M.







