

HY-N2150 · 100 g
MedChemExpress · Cat: HY-N2150
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Manufacturer product page
medchemexpress.com/psammaplin-a.html
Description
Psammaplin A is a marine metabolite. Psammaplin A is a selective HDAC1 IC50: 45 nM , DNA methyltransferases IC50: 18.6 nM and aminopeptidase N APN IC50: 18 ?M inhibitor. Psammaplin A also inhibits DNA topoisomerase and farnesyl protein transferase. Psammaplin A is a PPAR? activator and induces apoptosis. Psammaplin A has antitumor and anti-inflammatory activities. Psammaplin A has antibacterial activity against Gram-positive bacteria and inhibits DNA synthesis and DNA gyrase activity. Psammaplin A inhibits angiogenesis.







