

HY-163651 · 50 mg
MedChemExpress · Cat: HY-163651
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Manufacturer product page
medchemexpress.com/r-vorbipiprant.html
Description
R -Vorbipiprant R -CR6086 is an orally active antagonist for prostaglandin E2 receptor 4 EP4 with Ki of 16.6 nM for human EP4. R -Vorbipiprant inhibits PGE2 HY-101952 -induced cAMP production with an IC50 of 22 nM. R -Vorbipiprant exhibits immunomodulatory and anti-angiogenic activities, and ameliorates the collagen-induced arthritis in mice.







