

HY-16729A · Free Sample (0.1 - 0.2 mg)
MedChemExpress · Cat: HY-16729A
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medchemexpress.com/relenopride-hydrochloride.htmlDescription
Relenopride YKP10811 hydrochloride is a specific and selective 5-HT4 receptor agonist Ki=4.96 nM . Relenopride hydrochloride has 120-fold and 6-fold lower affinity, respectively, for 5-HT2A Ki=600 nM and 5-HT2B receptors Ki=31 nM than for 5-HT4. Relenopride hydrochloride increases gastrointestinal GI motility.







