

HY-114962 · 10 mM * 1 mL in DMSO
MedChemExpress · Cat: HY-114962
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Manufacturer product page
medchemexpress.com/s-22153.html
Description
S-22153 is a potent melatonin receptor antagonist with EC50 values of 19 nM, 4.6 nM for hMT1 and hMT2 melatonin receptor, respectively. S-22153 has Ki values of 8.6 nM CHO cells and 16.3 nM HEK cells for hMT1, and 6.0 nM CHO cells and 8.2 nM HEK cells for hMT2. S-22153 is a specific ligand of MT1 and MT2 melatonin receptors subtypes.







