GENERAL CATALOGUE
S1RA hydrochloride
HY-18099A · Free Sample (0.1 - 0.2 mg)
MedChemExpress · Cat: HY-18099A
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medchemexpress.com/S1RA-hydrochloride.htmlCatalog No: HY-18099A
CAS No: 1265917-14-3
Category: GPCR G Protein
Pack Size: Free Sample (0.1 - 0.2 mg)
Brand: MedChemExpress
Description
S1RA E-52862 hydrochloride is an orally active and selective sigma-1 receptor ?1R antagonist with a Ki value of 17 nM. S1RA hydrochloride shows good selectivity against ?2R Ki 1000 nM. S1RA hydrochloride is a human 5-HT2B receptor antagonist with an IC50 value of 4.7 ?M. S1RA hydrochloride inhibits neuropathic pain and activity-induced spinal sensitization.
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