

HY-P10819 · 50 mg
MedChemExpress · Cat: HY-P10819
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Manufacturer product page
medchemexpress.com/s9-cmc1-tfa.html
Description
S9-CMC1 TFA is a covalent peptide lysine-specific demethylase 1 LSD1 inhibitor with an IC50 value of 2.53 ?M. S9-CMC1 TFA specifically recognizes Cys360 in the enzyme-active region. S9-CMC1 TFA inhibits LSD1 activity, increasing H3K4me1 and H3K4me2 levels, leading to G1 cell cycle arrest and apoptosis and inhibiting cell proliferation. S9-CMC1 TFA significantly inhibits tumor growth in A549 xenograft animal models.







