Sarpogrelate-d3 hydrochloride

Description

Sarpogrelate-d3 hydrochloride is the deuterium labeled Sarpogrelate hydrochloride. Sarpogrelate hydrochloride MCI-9042 is a selective 5-HT2R antagonist, with pKis of 8.52, 6.57, and 7.43 for 5-HT2A, 5-HT2B, and 5-HT2C receptors, respectively. Sarpogrelate hydrochloride displays selectivity over 5-HT1, 5-HT3, 5-HT4, ?1-, ?2- and ?-adrenoreceptor, histamine H1, H2 and muscarinic M3 receptors. Sarpogrelate hydrochloride can be used for the research of vascular disease associated with thrombosis.