GENERAL CATALOGUE
SB-277011 hydrochloride
HY-10847B · Free Sample (0.1 - 0.2 mg)
MedChemExpress · Cat: HY-10847B
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medchemexpress.com/sb-277011-hydrochloride.htmlCatalog No: HY-10847B
CAS No: 215804-67-4
Category: GPCR G Protein
Pack Size: Free Sample (0.1 - 0.2 mg)
Brand: MedChemExpress
Description
SB-277011 hydrochloride SB-277011A hydrochloride is a potent, selective, orally bioavailable and brain penetrate dopamine D3 receptor D3R antagonist with Ki values of 10.7 nM and 11.2 nM at rodent and human D3R, respectively. SB-277011 hydrochloride displays 80- to 100-fold selectivity over other dopamine receptors with pKis of 8.0, 6.0, <5.2, and 5.9 for D3, D2, 5-HT1B, and 5-HT1D receptors, respectively.
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