

HY-161885 · 50 mg
MedChemExpress · Cat: HY-161885
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medchemexpress.com/smarca2-in-6.htmlDescription
SMARCA2-IN-6 is a SMARCA2 also known as BRM inhibitor, with IC50s less than 5 nM for SMARCA2 and SMARCA4. SMARCA2-IN-6 inhibits KRT80 gene expression in H1299 cells IC50: 26 nM . SMARCA2-IN-6 inhibits proliferation in BRG1-mutant SKMEL5 cells IC50: 13 nM .

