

HY-106756 · 50 mg
MedChemExpress · Cat: HY-106756
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medchemexpress.com/spiradoline.html
Description
Spiradoline U-62066 , an arylacetamide, is a selective kappa opioid receptor KOR agonist with a Ki of 8.6 nM in guinea pig. The Ki values of Spiradoline for ? and ? receptors are 252 nM and 9400 nM, respectively. Spiradoline has potent diuretic, analgesic, antiarrythmic, antitussive, neuroprotective properties and easily penetrates the blood-brain barrier.







