GENERAL CATALOGUE
TAK-683 TFA
HY-P2161A · 50 mg
MedChemExpress · Cat: HY-P2161A
Reach 3+ verified distributors
Manufacturer product page
medchemexpress.com/tak-683-tfa.html
Sponsored
Catalog No: HY-P2161A
Category: GPCR G Protein
Pack Size: 50 mg
Brand: MedChemExpress
Description
TAK-683 TFA is a potent full KISS1 receptor KISS1R agonist IC50=170 pM with improved metabolic stability. TAK-683 TFA is a nonapeptide metastin analog, exhibits agonistic activities to KISS1R with EC50 values of 0.96 nM and 1.6 nM for human and rat, respectively. TAK-683 TFA depletes GnRH in the hypothalamus and reduces plasma FSH, LH, and testosterone levels in vivo, it has the potential for the study of hormone-dependent prostate cancer.
More from MedChemExpress
GPR120 Agonist 1
HY-108711
GPCR G Protein
AG-045572
HY-107534
GPCR G Protein
Pamabrom
HY-17391
GPCR G Protein
ZD-7114
HY-101320
GPCR G Protein
Vasopressin Dimer (anti-parallel) (TFA)
HY-P5214
GPCR G Protein
Zimeldine-d6
HY-118835S
GPCR G Protein
ZM241385 (Standard)
HY-19532R
GPCR G Protein
(5S,6S)-DiHETE
HY-130138
GPCR G Protein