GENERAL CATALOGUE
TAN-452
HY-136208 · 10 mM * 1 mL in DMSO
MedChemExpress · Cat: HY-136208
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medchemexpress.com/tan-452.htmlCatalog No: HY-136208
CAS No: 892039-23-5
Category: GPCR G Protein
Pack Size: 10 mM * 1 mL in DMSO
Brand: MedChemExpress
Description
TAN-452 is an orally active, selective peripherally acting ?-opioid receptor DOR antagonist with a Ki of 0.47?nM and a Kb of 0.21?nM. TAN-452 is an antagonist for ?-opioid receptor MOR; Ki=36.56?nM and Kb=9.43?nM and ?-opioid receptor KOR; Ki=5.31?nM and Kb=7.18?nM . TAN-452, a derivative of Naltrindole, demonstrates low brain penetrability and attenuates morphine-induced side effects without affecting pain control.
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