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TCF4/?-catenin-IN-1
GENERAL CATALOGUE

TCF4/?-catenin-IN-1

HY-172393 · 50 mg

MedChemExpress · Cat: HY-172393

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Catalog No: HY-172393
Category: Apoptosis
Pack Size: 50 mg
Brand: MedChemExpress

Description

TCF4/?-catenin-IN-1 Compound 8b is an inhibitor of TCF4/?-catenin, and induces apoptosis. TCF4/?-catenin-IN-1 up-regulates p53, caspase-3, caspase-8, caspase-9 levels and Bax protein expression as well as down-regulates Bcl-2 protein expression. TCF4/?-catenin-IN-1 can inhibit CYP3A4, CYP1A2, CYP2C19, and shows promising cytotoxic activity in cancer cells.

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