

HY-172393 · 50 mg
MedChemExpress · Cat: HY-172393
Reach 3+ verified distributors
Manufacturer product page
medchemexpress.com/tcf4-%CE%B2-catenin-in-1.html
Description
TCF4/?-catenin-IN-1 Compound 8b is an inhibitor of TCF4/?-catenin, and induces apoptosis. TCF4/?-catenin-IN-1 up-regulates p53, caspase-3, caspase-8, caspase-9 levels and Bax protein expression as well as down-regulates Bcl-2 protein expression. TCF4/?-catenin-IN-1 can inhibit CYP3A4, CYP1A2, CYP2C19, and shows promising cytotoxic activity in cancer cells.







