GENERAL CATALOGUE
Theliatinib tartrate
HY-104066A · 50 mg
MedChemExpress · Cat: HY-104066A
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Manufacturer product page
medchemexpress.com/theliatinib-tartrate.htmlCatalog No: HY-104066A
CAS No: 2413487-72-4
Category: JAK STAT Signaling
Pack Size: 50 mg
Brand: MedChemExpress
Description
Theliatinib Xiliertinib tartrate is a potent, ATP-competitive, orally active and highly selective EGFR inhibitor with a Ki of 0.05 nM and an IC50 of 3 nM. Theliatinib has an IC50 of 22 nM for EGFR T790M/L858R mutant. Theliatinib shows >50-fold selectivity for EGFR than other kinases. Theliatinib tartrate is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition CuAAc with molecules containing Azide groups.
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