

HY-B1213A · 50 mg
MedChemExpress · Cat: HY-B1213A
Reach 3+ verified distributors
Manufacturer product page
medchemexpress.com/trimipramine.html
Description
Trimipramine is a 5-HT receptor antagonist, with pKi binding values of 6.39, 8.10, 4.66 for 5-HT1C, 5-HT2 and 5-HT1A, respectively. Trimipramine is also a potent and selective inhibitor targeting human noradrenaline hNAT , serotonin hSERT and organic cation transporters hOCT1, hOCT2 with IC50 values of 4.99 ?M, 2.11 ?M, 3.72 ?M, 8.00 ?M, respectively. Trimipramine has vascular activity and anxiolytic efficacy.