Trimipramine (Standard)

Description

Trimipramine Standard is the analytical standard of Trimipramine. This product is intended for research and analytical applications. Trimipramine is a 5-HT receptor antagonist, with pKi binding values of 6.39, 8.10, 4.66 for 5-HT1C, 5-HT2 and 5-HT1A, respectively. Trimipramine is also a potent and selective inhibitor targeting human noradrenaline hNAT , serotonin hSERT and organic cation transporters hOCT1, hOCT2 with IC50 values of 4.99 ?M, 2.11 ?M, 3.72 ?M, 8.00 ?M, respectively. Trimipramine has vascular activity and anxiolytic efficacy.