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TrimTAC1
GENERAL CATALOGUE

TrimTAC1

HY-169355 · 50 mg

MedChemExpress · Cat: HY-169355

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medchemexpress.com/trimtac1.html
Catalog No: HY-169355
CAS No: 3095569-91-5
Category: Epigenetics
Pack Size: 50 mg
Brand: MedChemExpress

Description

TrimTAC1 is a TRIM21-based PROTAC targeting BRD4. TrimTAC1 selectively degrads NUP98FG-mEGFP-BRD4BD2 nuclear condensates. TrimTAC1 does not degrade soluble mEGFP-BRD4BD2 in A549 cells. Pink: target protein ligand + -JQ-1 HY-13030 ; Blue:E3 ligase ligand Acepromazine-OTs HY-169356 ; Black: PROTAC linker HY-W088456 ; E3 ligase ligand + linker: HY-169357 .

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