

HY-169355 · 50 mg
MedChemExpress · Cat: HY-169355
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Manufacturer product page
medchemexpress.com/trimtac1.html
Description
TrimTAC1 is a TRIM21-based PROTAC targeting BRD4. TrimTAC1 selectively degrads NUP98FG-mEGFP-BRD4BD2 nuclear condensates. TrimTAC1 does not degrade soluble mEGFP-BRD4BD2 in A549 cells. Pink: target protein ligand + -JQ-1 HY-13030 ; Blue:E3 ligase ligand Acepromazine-OTs HY-169356 ; Black: PROTAC linker HY-W088456 ; E3 ligase ligand + linker: HY-169357 .







