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TRPM8 antagonist 4
GENERAL CATALOGUE

TRPM8 antagonist 4

HY-174825 · 50 mg

MedChemExpress · Cat: HY-174825

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Catalog No: HY-174825
Category: Apoptosis
Pack Size: 50 mg
Brand: MedChemExpress

Description

TRPM8 antagonist 4 is a CB2R partial agonist EC50=54.2 nM, Ki=3.2 ?M and TRPM8 antagonists IC50=42.3 nM with high functional selectivity and good physicochemical properties. TRPM8 antagonist 4 has significant anti-inflammatory and analgesic effects and good safety, reduces the mRNA expression of TNF-?, IL-6, and IL-1?.

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