GENERAL CATALOGUE
TRPV1 antagonist 11
HY-176063 · 50 mg
MedChemExpress · Cat: HY-176063
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medchemexpress.com/trpv1-antagonist-11.htmlCatalog No: HY-176063
CAS No: 3084843-71-7
Category: GPCR G Protein
Pack Size: 50 mg
Brand: MedChemExpress
Description
TRPV1 antagonist 11 compound 2ac is a potent TRPV1 antagonist with an IC50 of 29.3 nM. TRPV1 antagonist 11 is a potent ?-opioid receptor MOR agonist with a Ki of 60.3 nM. TRPV1 antagonist 11, a pyrimidine piperazine, exhibits pain relieving effects by antagonizing TRPV1 and stimulating MOR. TRPV1 antagonist 11 shows a potent, dose-dependent anti-nociceptive effect in a Formalin-induced pain model in mice.
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