

HY-N2346 · 5 mg
MedChemExpress · Cat: HY-N2346
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Manufacturer product page
medchemexpress.com/tubulysin-e.html
Description
Tubulysin E is a highly cytotoxic anti-microtubule toxin anti-microtubule toxins that is synthesized as an ADC cytotoxin ADC Cytotoxin . Tubulysin E can be isolated from the myxobacteria Archangium geophyra and Angiococcus disciformis. Tubulysin E displays extremely potent cytotoxic activity in mammalian cells, including multidrug-resistant cell lines, with IC50 values in the low nanomolar range. Tubulysin E inhibits microtubule/Tubulin polymerization and leads to cell cycle arrest and apoptosis.







