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Tubulysin E
GENERAL CATALOGUE

Tubulysin E

HY-N2346 · 5 mg

MedChemExpress · Cat: HY-N2346

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medchemexpress.com/tubulysin-e.html
Catalog No: HY-N2346
CAS No: 309935-58-8
Category: Antibody-drug Conjugate ADC Related
Pack Size: 5 mg
Brand: MedChemExpress

Description

Tubulysin E is a highly cytotoxic anti-microtubule toxin anti-microtubule toxins that is synthesized as an ADC cytotoxin ADC Cytotoxin . Tubulysin E can be isolated from the myxobacteria Archangium geophyra and Angiococcus disciformis. Tubulysin E displays extremely potent cytotoxic activity in mammalian cells, including multidrug-resistant cell lines, with IC50 values in the low nanomolar range. Tubulysin E inhibits microtubule/Tubulin polymerization and leads to cell cycle arrest and apoptosis.

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