

HY-12279A · 50 mg
MedChemExpress · Cat: HY-12279A
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medchemexpress.com/umbralisib-tosylate.htmlDescription
Umbralisib TGR-1202 tosylate is an orally active, potent and selective dual PI3K? and casein kinase-1-? CK1? inhibitor, with EC50 of 22.2 nM and 6.0 ?M, respectively. Umbralisib tosylate exhibits unique immunomodulatory effects on chronic lymphocytic leukemia CLL T cells. Umbralisib tosylate can be used for haematological malignancies reseach.