

HY-173156 · 5 mg
MedChemExpress · Cat: HY-173156
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Manufacturer product page
medchemexpress.com/unc10013.html
Description
UNC10013 is a SETDB1 allosteric modulator that forms a covalent bond with Cys385 in the 3TD domain, exhibiting negative allosteric regulatory activity. It has a kinact/KI value of 1.0 AAAasAa 106 M-1s-1. UNC10013 effectively disrupts SETDB1-mediated Akt methylation and holds potential value for research in cancer and neurodegenerative diseases.

