

HY-W727879 · 1 mg
MedChemExpress · Cat: HY-W727879
Reach 3+ verified distributors
Manufacturer product page
medchemexpress.com/upadacitinib-15n-d2.htmlDescription
Upadacitinib-15N,d2 ABT-494-15N,d2 is the deuterium-labeled Upadacitinib HY-19569 . Upadacitinib-15N,d2 ABT-494 is a potent, orally active and selective Janus kinase 1 JAK1 inhibitor IC50=43 nM . Upadacitinib-15N,d2 ABT-494 displays approximately 74 fold selective for JAK1 over JAK2 200 nM in cellular assays dependent on specific, relevant cytokines. Upadacitinib-15N,d2 ABT-494 can be used for several autoimmune disorders research.