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XYD190
GENERAL CATALOGUE

XYD190

HY-161494 · 50 mg

MedChemExpress · Cat: HY-161494

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Manufacturer product page

medchemexpress.com/xyd190.html
Catalog No: HY-161494
Category: Epigenetics
Pack Size: 50 mg
Brand: MedChemExpress

Description

XYD190 Compound 14g is an orally active degrader for CBP/p300. XYD190 inhibits CBP/p300 bromodomain with IC50 of 483.7 nM. XYD190 exhibits antitumor activity against acute myeloid leukemia. Structure: Pink, CBP/p300 ligand 4 HY-161495 ; Blue, E3 ligase ligand HY-14658 ; Black: linker HY-161496 .

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